Product Description
| Cat Number | T15286 |
|---|---|
| Category | Biochemical |
| Pack Size | 1EA |
| Description | Flindokalner (BMS-204352) is a potassium channel modulator and a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. It is also a positive modulator of large conductance calcium-activated K channels (BKca) and displays negative modulatory activity at Kv7.1 channels (Ki = 3.7 μM). Additionally, Flindokalner acts as a negative modulator of GABAA receptors and demonstrates anxiolytic efficacy in vivo. |
| Molecular Weight | 359.7 |
| Purity | 0.9925 |
| Formula | C16H10ClF4NO2 |
| Smiles | COc1ccc(Cl)cc1[C@]1(F)C(=O)Nc2cc(ccc12)C(F)(F)F |
| Storage | -20 ℃ |
| View Document | |
| Note | This product is for Research Use Only |

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