Product Description
| Cat Number | T17243 |
|---|---|
| Category | Biochemical |
| Pack Size | 1EA |
| Description | VU0463271 (N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide) is a potent and selective antagonist of the neuronal-specific potassium-chloride cotransporter 2 (KCC2), with an IC50 of 61 nM and >100-fold selectivity versus the closely related Na-K-2Cl cotransporter 1 (NKCC1) and no activity in a larger panel of GPCRs, ion channels, and transporters. |
| Molecular Weight | 382.5 |
| Purity | 0.9975 |
| Formula | C19H18N4OS2 |
| Smiles | Cc1csc(n1)N(C1CC1)C(=O)CSc1ccc(nn1)-c1ccccc1 |
| Storage | -20 ℃ |
| View Document | |
| Note | This product is for Research Use Only |
Share Item: