Product Description
| Cat Number | T25310 |
|---|---|
| Category | Biochemical |
| Pack Size | 1EA |
| Description | Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14, and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m), and rat (r) MC1R, respectively. Dersimelagon exhibits good affinity for hMC1R and hMC4R, with Ki values of 2.26 and 32.9 nM, respectively. Dersimelagon can be used in the study of skin pigmentation[1]. |
| Molecular Weight | 675.75 |
| Purity | 0.9823 |
| Formula | C36H45F4N3O5 |
| Smiles | C(=O)([C@@]1(F)[C@@H](CN(C1)C2CCCC2)C3=CC=C(OC)C=C3)N4C[C@@H]([C@@H](COC)C4)C5=C(C=C(C(F)(F)F)C=C5)N6CCC(C(O)=O)CC6 |
| Storage | -20 ℃ |
| View Document | |
| Note | This product is for Research Use Only |
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