Product Description
| Cat Number | T29231 |
|---|---|
| Category | Biochemical |
| Pack Size | 1EA |
| Description | ZLD1039 is a potent, orally bioavailable EZH2 (Enhancer of Zeste Homolog 2) inhibitor with high selectivity. It demonstrates strong, concentration-dependent inhibition of both wild-type and mutant (Y641F and A677G) PRC2 (Polycomb Repressive Complex 2) enzymatic activities, exhibiting IC50 values of 5.6, 15, and 4.0 nM, respectively. Additionally, ZLD1039 effectively suppresses breast tumor growth and metastasis. |
| Molecular Weight | 612.8 |
| Purity | 0.9982 |
| Formula | C36H48N6O3 |
| Smiles | CCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c3CCCCc3c(C)[nH]c2=O)c1C)-c1ccc(nc1)N1CCN(C)CC1 |
| Storage | -20 ℃ |
| View Document | |
| Note | This product is for Research Use Only |
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