Product Description
| Cat Number | T3624 |
|---|---|
| Category | Biochemical |
| Pack Size | 1EA |
| Description | A-366 is a highly selective peptide-competitive histone methyltransferase G9a inhibitor with IC50s of 3.3 and 38 nM for G9a and GLP, respectively.It is more than 1,000-fold selective for G9a and GLP over the other 21 methyltransferases. It is an inhibitor of the Spindlin1-H3K4me3 interaction with an IC50 of 182.6 nM.It exhibits high affinity for human H3R with a Ki value of 17 nM, and shows subtype selectivity between subgroups of the histaminergic and dopaminergic receptor families. |
| Molecular Weight | 329.44 |
| Purity | 0.9853 |
| Formula | C19H27N3O2 |
| Smiles | COc1cc2c(cc1OCCCN1CCCC1)N=C(N)C21CCC1 |
| Storage | -20 ℃ |
| View Document | |
| Note | This product is for Research Use Only |
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